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Information

AHFS Class:

28:08.12 Opiate Partial Agonists


Generic Name

Products

Nalbuphine hydrochloride is available as a 10- or 20-mg/mL solution in 1-mL ampuls and 10-mL multiple-dose vials.997 Each mL contains nalbuphine hydrochloride 10 or 20 mg, sodium citrate dihydrate 0.47 mg, and citric acid anhydrous 0.63 mg with sodium hydroxide and/or hydrochloric acid for pH adjustment and sodium chloride for tonicity.997 Multiple-dose vials also contain, in each mL, methylparaben 1.8 mg and propylparaben 0.2 mg as preservatives.997

pH

From 3 to 4.5.997

Administration

Nalbuphine hydrochloride is administered by subcutaneous, intramuscular, or intravenous injection.997

Stability

Intact vials and ampuls should be stored at controlled room temperature and protected from excessive light.997 Ampuls should be kept in the ampul tray until time of use and unused portions should be discarded.997 Multiple-dose vials should be retained in the carton until contents are used.997

Central Venous Catheter

Nalbuphine hydrochloride (Astra) 1 mg/mL in dextrose 5% was found to be compatible with the ARROWg+ard Blue Plus (Arrow International) chlorhexidine-bearing triple-lumen central catheter. Essentially complete delivery of the drug was found with little or no drug loss occurring. Furthermore, chlorhexidine delivered from the catheter remained at trace amounts with no substantial increase due to the delivery of the drug through the catheter.2335

Compatibility

Solution Compatibility

Drugs in Syringe Compatibility

Y-Site Injection Compatibility (1:1 Mixture)

Other Info

References

For a list of references cited in the text of this monograph, search the monograph titled References.

Copyrights

ASHP® Injectable Drug InformationTM. Selected Revisions March 31, 2024. © Copyright, 2024. American Society of Health-System Pharmacists®, 4500 East-West Highway, Suite 900, Bethesda, Maryland 20814.