Contraindicated in:
Use Cautiously in:
CNS: headache.
CV: HF, edema, hypotension, tachycardia, palpitations.
Derm: hirsutism, rash.
Endo: DIABETIC KETOACIDOSIS, HYPEROSMOLAR NONKETOTIC COMA, hyperglycemia, hyperuricemia.
GI: ILEUS, abdominal pain, diarrhea, loss of taste, nausea, vomiting.
GU: glycosuria.
Hemat: neutropenia, thrombocytopenia.
Resp: PULMONARY HYPERTENSION.
MS: weakness.
Drug-Drug:
Drug-Natural Products:
(Generic available)
Hyperinsulinemic Hypoglycemia
Absorption: Well absorbed following oral administration.
Distribution: Crosses the blood-brain barrier and placenta.
Protein Binding: >90%.
Metabolism/Excretion: 50% metabolized by the liver; 50% excreted unchanged by the kidneys.
Half-life: 1036 hr (↑ in renal impairment).