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Indications

REMS

Contraind./Precautions

Contraindicated in:

Use Cautiously in:

Exercise Extreme Caution in:

Adv. Reactions/Side Effects

CV: ECG changes, angina, chest tightness/pressure, coronary vasospasm, MI, transient hypertension, VENTRICULAR FIBRILLATION, VENTRICULAR TACHYCARDIA.

GI: abdominal pain, dry mouth, dysphagia, nausea.

Neuro: dizziness, drowsiness, paresthesia, weakness.
Misc: ANAPHYLAXIS.

Interactions

Drug-Drug:

Availability

(Generic available)

Route/Dosage

US Brand Names

Relpax

Action

Therapeutic Effects:

Classifications

Therapeutic Classification: vascular headache suppressants

Pharmacologic Classification: five ht1 agonists

Pharmacokinetics

Absorption: 50% absorbed after oral administration.

Distribution: Enters breast milk.

Metabolism/Excretion: Mostly metabolized by the liver via the CYP3A4 enzyme system.

Half-life: 4 hr.

Time/Action Profile

(decreased migraine pain)

ROUTEONSETPEAKDURATION
POwithin 2 hr2 hrup to 24 hr

Patient/Family Teaching

Pronunciation

e-le-TRIP-tan