section name header

Pronunciation

al-BYOO-ter-ole

Classifications

Therapeutic Classification: bronchodilators

Pharmacologic Classification: adrenergics

Indications

REMS

Action

Therapeutic Effects:

Pharmacokinetics

Absorption: Well absorbed after oral administration but rapidly undergoes extensive metabolism.

Distribution: Small amounts appear in breast milk.

Metabolism/Excretion: Extensively metabolized by the liver and other tissues.

Half-life: Oral 2.7–5 hr; Inhalation: 3.8 hr.

Time/Action Profile

(bronchodilation)

ROUTEONSETPEAKDURATION
PO15–30 min2–3 hr4–6 hr or more
Inhaln5–15 min60–90 min3–6 hr

Contraind./Precautions

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects

CV: chest pain, palpitations, angina, arrhythmias, hypertension.

Endo: hyperglycemia.

F and E: hypokalemia.

GI: nausea, vomiting.

Neuro: nervousness, restlessness, tremor, headache, hyperactivity (children), insomnia.

Resp: PARADOXICAL BRONCHOSPASM (EXCESSIVE USE OF INHALERS).

Interactions

Drug-Drug:

Drug-Natural Products:

Route/Dosage

see Calculator

Availability

(Generic available)

Assessment

Lab Test Considerations:

Implementation

Patient/Family Teaching

Evaluation/Desired Outcomes

US Brand Names

Accuneb, Proair Digihaler, Proair HFA, Proair Respiclick, Proventil HFA, Ventolin HFA, VoSpire ER

Canadian Brand Names

Airomir, Salbutamol, Ventolin Diskus, Ventolin Nebules

Pill Image

albuterol_sulfate_195_9142.jpg

Code

NDC Code*