Contraindicated in:
Use Cautiously in:
CNS: asthenia.
Derm: alopecia.
GI: abdominal pain, ↓ appetite, diarrhea, nausea, vomiting, stomatitis.
Hemat: anemia, neutropenia, THROMBOCYTOPENIA.
Misc: fever.
Absorption: Well absorbed following oral administration.
Distribution: Unknown.
Protein Binding: Trifluridine >96%.
Metabolism/Excretion: Trifluridine is metabolized by thymidine phosphorylase to an inactive metabolite. Trifluridine 1.5% excreted unchanged in urine; tipiracil 29.3% excreted unchanged in urine.
Half-life: Trifluridine 2.1 hr; tipiracil 2.4 hr.
NDC Code*