Contraindicated in:
Use Cautiously in:
CV: hypotension, palpitations.
Derm: photosensitivity.
EENT: blurred vision, tinnitus.
GI: anorexia, constipation, diarrhea, dry mouth.
GU: dysuria, urinary frequency.
Local: pain at IM site.
Neuro: drowsiness, dizziness, headache, paradoxical excitation (children).
Drug-Drug:
(Generic available)
Absorption: Well absorbed after oral or IM administration. IV administration results in complete bioavailability.
Distribution: Extensively distributed to tissues.
Metabolism/Excretion: Metabolized by the liver.
Half-life: Unknown.
(antimotion sickness, antiemetic activity)
ROUTE | ONSET | PEAK | DURATION |
---|---|---|---|
PO | 1560 min | 12 hr | 36 hr |
IM | 2030 min | 12 hr | 36 hr |
IV | rapid | unknown | 36 hr |
NDC Code*