Contraindicated in:
Use Cautiously in:
CV: chest pain, edema, palpitations, COMPLETE HEART BLOCK, HF, MI, angina, atrial fibrillation, CEREBROVASCULAR ACCIDENT, orthostatic hypotension, pericardial effusion, pericarditis, tachycardia, TORSADE DE POINTES, VENTRICULAR TACHYCARDIA.
Derm: alopecia, pruritus, rash.
EENT: abnormal vision.
GI: abdominal pain, diarrhea, flatulence, GI BLEEDING, anorexia, constipation, dyspepsia, HEPATOTOXICITY, nausea, PANCREATITIS, vomiting.
GU: dysuria, ↓ fertility (females), hematuria, RENAL FAILURE.
Hemat: anemia.
MS: weakness, arthralgia, back pain, myalgia.
Neuro: dizziness, headache, malaise, paresthesia , SEIZURES.
Resp: dyspnea, cough, EOSINOPHILIC PNEUMONIA, INTERSTITIAL PNEUMONITIS, pharyngitis, PULMONARY FIBROSIS, PULMONARY HYPERTENSION.
Misc: fever.
Drug-Drug:
Hepatic Impairment
Absorption: Well absorbed after oral administration.
Distribution: Unknown.
Metabolism/Excretion: Extensively metabolized; <1% excreted unchanged in urine.
Half-life: 1.3 hr.
(↓ in platelet count)
ROUTE | ONSET | PEAK | DURATION |
---|---|---|---|
PO | 714 days | 412 wk | 4 days |
Increase in platelet count after discontinuation.
NDC Code*