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Indications

REMS

Contraind./Precautions

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects

F and E: LACTIC ACIDOSIS.

GI: abdominal bloating, diarrhea, nausea, vomiting, unpleasant metallic taste.

Hemat: ↓ vitamin B12 levels.

Interactions

Drug-Drug:

Drug-Natural Products:

Availability

(Generic available)

Route/Dosage

US Brand Names

Glucophage XR, Glumetza, Riomet, Riomet ER

Action

Therapeutic Effects:

Classifications

Therapeutic Classification: antidiabetics

Pharmacologic Classification: biguanides

Pharmacokinetics

Absorption: 50–60% absorbed after oral administration.

Distribution: Extensively distributed to tissues.

Metabolism/Excretion: Eliminated almost entirely unchanged by the kidneys.

Half-life: 17.6 hr.

Canadian Brand Names

Glucophage, Glycon

Time/Action Profile

(plasma concentrations)

ROUTEONSETPEAKDURATION
PO-IRunknownunknown12 hr
PO-ERunknown4–8 hr24 hr

Patient/Family Teaching

Pronunciation

met-FOR-min audio

Pill Image

metforminhcl_195_8795.jpg

Code

NDC Code*