Contraindicated in:
Use Cautiously in:
Derm: rash, photosensitivity, pruritus.
GI: HEPATOTOXICITY, abdominal pain, anorexia, gastrointestinal reflux disease, nausea, diarrhea, dyspepsia, vomiting, weight loss, dysgeusia.
MS: arthralgia.
Drug-Drug:
Absorption: Absorption follows oral administration. Food ↓ rate and extent of absorption.
Distribution: Unknown.
Metabolism/Excretion: Mostly metabolized by the CYP1A2 enzyme system, some metabolism by other CYP enzymes. 80% excreted in urine as inactive metabolite.
Half-life: 3 hr.
NDC Code*