Canada-Approved Medicine
This monograph describes a medication approved for use in Canada by the Therapeutic Products Directorate, a division of Health Canadas Health Products and Food Branch. The medication is not approved by the United States Food and Drug Administration; however, a similar formulation carrying a different generic or brand name might be available in the US.
REMSContraindicated in:
Use Cautiously in:
CNS: headache, dizziness, fatigue.
CV: palpitations, ↓ PR interval, tachycardia.
GI: abdominal pain, diarrhea, nausea, vomiting.
Drug-Drug:
Renal Impairment
Therapeutic Classification: prokinetic agents
Pharmacologic Classification: dihydrobenzofurancarboxamides
Absorption: Rapidly absorbed (90%) following oral administration.
Distribution: Rapidly and extensively distributed, enters breast milk.
Metabolism/Excretion: 60% excreted unchanged in urine, 38% unchanged in feces, minor amounts are extensively metabolized.
Half-life: 24 hr.