section name header

Indications ⬇

BEERS REMS

Unlabeled Use:

Contraind./Precautions ⬆ ⬇

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects ⬆ ⬇

CV: QT interval prolongation, hypotension, tachycardia, TORSADES DE POINTES, ventricular arrhythmias.

Derm: diaphoresis, photosensitivity, rash.

EENT: blurred vision, dry eyes.

Endo: amenorrhea, galactorrhea, gynecomastia.

GI: constipation, dry mouth, anorexia, hepatitis, ileus.

GU: impotence, urinary retention.

Hemat: AGRANULOCYTOSIS, anemia, leukopenia, neutropenia.

Metab: weight gain.

Neuro: extrapyramidal reactions, confusion, drowsiness, restlessness, SEIZURES, tardive dyskinesia.

Resp: respiratory depression.

Misc: hypersensitivity reactions, NEUROLEPTIC MALIGNANT SYNDROME.

Interactions ⬆ ⬇

Drug-Drug:

Drug-Natural Products:

Availability ⬆ ⬇

(Generic available)

Route/Dosage ⬆ ⬇

see Calculator

Haloperidol

Haloperidol Decanoate

US Brand Names ⬆ ⬇

Haldol, Haldol Decanoate

Action ⬆ ⬇

Therapeutic Effects:

Classifications ⬆ ⬇

Therapeutic Classification: antipsychotics

Pharmacologic Classification: butyrophenones

Pharmacokinetics ⬆ ⬇

Absorption: Well absorbed following PO/IM administration. Decanoate salt is slowly absorbed and has a long duration of action.

Distribution: Concentrates in liver.

Protein Binding: 92%.

Metabolism/Excretion: Mostly metabolized by the liver.

Half-life: 21–24 hr.

Time/Action Profile ⬆ ⬇

(antipsychotic activity)

ROUTEONSETPEAKDURATION
PO2 hr2–6 hr8–12 hr
IM20–30 min30–45 min4–8 hr†
IM (decanoate)3–9 daysunknown1 mo

†Effect may persist for several days.

Patient/Family Teaching ⬆ ⬇

Pronunciation ⬆ ⬇

ha-loe-PER-i-dole audio

Code ⬆

NDC Code*