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Indications

REMS

Contraind./Precautions

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects

F and E: hypokalemia (with chronic use).

GI: abdominal cramps, nausea, diarrhea, rectal burning.

MS: muscle weakness (with chronic use).

Misc: protein-losing enteropathy, tetany (with chronic use).

Interactions

Drug-Drug:

Drug-Food:

Availability

(Generic available)

Route/Dosage

US Brand Names

Dulcolax, Ex-Lax Ultra

Action

Therapeutic Effects:

Classifications

Therapeutic Classification: laxatives

Pharmacologic Classification: stimulant laxatives

Pharmacokinetics

Absorption: Variable absorption follows oral administration; rectal absorption is minimal; action is local in the colon.

Distribution: Small amounts of metabolites excreted in breast milk.

Metabolism/Excretion: Small amounts absorbed are metabolized by the liver.

Half-life: Unknown.

Time/Action Profile

(evacuation of bowel)

ROUTEONSETPEAKDURATION
PO6–12 hrunknownunknown
Rectal15–60 minunknownunknown

Patient/Family Teaching

Pronunciation

bis-a-KOE-dill audio

Code

NDC Code*