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Indications ⬇

REMS


Unlabeled Use:

Contraind./Precautions ⬆ ⬇

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects ⬆ ⬇

CV: edema

F and E: metabolic alkalosis, hypernatremia, hypocalcemia, hypokalemia

GI: POflatulence, gastric distention

Local: irritation at IV site

Neuro: cerebral hemorrhage (with rapid injection in infants), tetany

Interactions ⬆ ⬇

Drug-drug:

Availability ⬆ ⬇

(Generic available)

Route/Dosage ⬆ ⬇

Alkalinization of Urine

Antacid

Systemic Alkalinization/Cardiac Arrest

Renal Tubular Acidosis

Action ⬆ ⬇

  • Acts as an alkalinizing agent by releasing bicarbonate ions.
  • Following oral administration, releases bicarbonate, which is capable of neutralizing gastric acid.
Therapeutic effects:
  • Alkalinization.
  • Neutralization of gastric acid.

Classifications ⬆ ⬇

Therapeutic Classification: antiulcer agents

Pharmacologic Classification: alkalinizing agents

Pharmacokinetics ⬆ ⬇

Absorption: Following oral administration, excess bicarbonate is absorbed, resulting in metabolic alkalosis and alkaline urine. IV administration results in complete bioavailability.

Distribution: Widely distributed into extracellular fluid.

Metabolism/Excretion: Sodium and bicarbonate are excreted by the kidneys.

Half-Life: Unknown.

Time/Action Profile ⬆ ⬇

( PO = antacid effect; IV = alkalinization)

ROUTEONSETPEAKDURATION
POimmediate30 min1–3 hr
IVimmediaterapidunknown

Patient/Family Teaching ⬆ ⬇

Pronunciation ⬆ ⬇

SOE-dee-um bye-KAR-boe-nate

Code ⬆

NDC Code