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Pronunciation

kloe-TRIM-a-zole

Indications

REMS

Action

Therapeutic Effects:

Pharmacokinetics

Absorption: Minimal systemic absorption.

Distribution: Inhibitory concentrations remain in saliva for up to 3 hr after troche dissolves.

Metabolism/Excretion: Metabolized by liver; <1% excreted unchanged in urine.

Half-life: 24 hr.

Contraind./Precautions

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects

GI: abnormal mouth sensations, liver function tests, nausea, vomiting.

Derm: pruritis.

Interactions

Drug-Drug:

Route/Dosage

Implementation

US Brand Names

Mycelex

Classifications

Therapeutic Classification: antifungals (oral, nonabsorbed)

Availability

(Generic available)

Time/Action Profile

ROUTEONSETPEAKDURATION
POunknownunknownup to 3 hr

Assessment

Lab Test Considerations:

Pot. Nursing Diagnoses

Patient/Family Teaching

Evaluation/Desired Outcomes

Code

NDC Code*