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Indications ⬇

REMS

Contraind./Precautions ⬆ ⬇

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects ⬆ ⬇

GI: abnormal mouth sensations, ↑ liver function tests, nausea, vomiting.

Derm: pruritis.

Interactions ⬆ ⬇

Drug-Drug:

Availability ⬆ ⬇

(Generic available)

Route/Dosage ⬆ ⬇

US Brand Names ⬆ ⬇

Mycelex

Action ⬆ ⬇

Therapeutic Effects:

Classifications ⬆ ⬇

Therapeutic Classification: antifungals (oral, nonabsorbed)

Pharmacokinetics ⬆ ⬇

Absorption: Minimal systemic absorption.

Distribution: Inhibitory concentrations remain in saliva for up to 3 hr after troche dissolves.

Metabolism/Excretion: Metabolized by liver; <1% excreted unchanged in urine.

Half-life: 24 hr.

Time/Action Profile ⬆ ⬇

ROUTEONSETPEAKDURATION
POunknownunknownup to 3 hr

Patient/Family Teaching ⬆ ⬇

Pronunciation ⬆ ⬇

kloe-TRIM-a-zole

Code ⬆

NDC Code*