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Indications

BEERS REMS

Contraind./Precautions

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects

EENT: blurred vision.

GI: dry mouth.

Neuro: drowsiness, fatigue.

Interactions

Drug-Drug:

Availability

(Generic available)

Route/Dosage

US Brand Names

Antivert, Bonine

Action

Therapeutic Effects:

Classifications

Therapeutic Classification: antiemetics, antihistamines

Pharmacokinetics

Absorption: Absorbed after oral administration.

Distribution: Unknown.

Metabolism/Excretion: Primarily metabolized by liver via the CYP2D6 isoenzyme; the CYP2D6 isoenzyme exhibits genetic polymorphism (7% of population may be poor metabolizers and may have significantly ↑ meclizine concentrations and an ↑ risk of adverse effects).

Half-life: 6 hr.

Time/Action Profile

(antihistaminic effects)

ROUTEONSETPEAKDURATION
PO1 hrunknown8–24 hr

Patient/Family Teaching

Pronunciation

MEK-li-zeen audio

Code

NDC Code*