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Indications ⬇

REMS

Contraind./Precautions ⬆ ⬇

Contraindicated in:

Use Cautiously in:

Adv. Reactions/Side Effects ⬆ ⬇

CV: chest pain, hypertension, peripheral edema.

Derm: hot flashes, alopecia, photosensitivity, rash, sweating.

Endo: breast pain, gynecomastia, hyperglycemia.

GI: constipation, diarrhea, nausea, ↑ liver enzymes, abdominal pain, HEPATOTOXICITY, vomiting.

GU: ↓ fertility, erectile dysfunction, hematuria, incontinence, nocturia, urinary tract infections.

Hemat: anemia.

Metab: ↓ weight.

MS: pain.

Neuro: weakness, dizziness, headache, insomnia, paresthesia.

Resp: dyspnea.

Misc: flu-like syndrome, infection.

Interactions ⬆ ⬇

Drug-Drug:

Availability ⬆ ⬇

(Generic available)

Route/Dosage ⬆ ⬇

US Brand Names ⬆ ⬇

Casodex

Action ⬆ ⬇

Therapeutic Effects:

Classifications ⬆ ⬇

Therapeutic Classification: antineoplastics

Pharmacologic Classification: antiandrogens

Pharmacokinetics ⬆ ⬇

Absorption: Well absorbed following oral administration.

Distribution: Unknown.

Protein Binding: 96%.

Metabolism/Excretion: Mostly metabolized by the liver. Excreted in the urine and feces.

Half-life: 5.8 days.

Time/Action Profile ⬆ ⬇

(plasma concentrations)

ROUTEONSETPEAKDURATION
POunknown31.3 hrunknown

Patient/Family Teaching ⬆ ⬇

Pronunciation ⬆ ⬇

bye-ka-LOOT-a-mide audio

Code ⬆

NDC Code*